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產(chǎn)品基本信息
產(chǎn)品編號:V128622
產(chǎn)品名稱:Vernakalant-d6 Hydrochloride
產(chǎn)品CAS:866455-16-5
規(guī)格含量:10mg
產(chǎn)品價格:面議
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產(chǎn)品詳細(xì)介紹
標(biāo)準(zhǔn)品編號:
V128622
名稱:
Vernakalant-d6 Hydrochloride
別名:
Vernakalant bis(Methoxy-d3) Hydrochloride; (3R)- 1-[(1R,2R)-2-[2-(3,4-Di(methoxy-d3)phenyl)ethoxy]cyclohexyl]-3-pyrrolidinol Hydrochloride; (1R,2R)-2-((3R)-Hydroxypyrrolidinyl)-1-(3,4-di(methoxy-d3)phenethoxy)cyclohexane Monohydrochloride; (1R,2R)-2-((3R)-Hydroxypyrrolidinyl)-1-[2-(3,4-di(methoxy-d3)phenyl)ethoxy]cyclohexane Monohydrochloride; (3R)-1-[(1R,2R)-2-[2-(3,4-Di(methoxy-d3)phenyl)ethoxy]cyclohexyl]-3-pyrrolidinol Monohydrochloride; RSD 1235-d3
CAS號:
866455-16-5
參考CAS號:
類似: 748810-28-8; free base: 866525-69-1
分子式:
C??H??D?ClNO?
分子量:
391.96
類別:
Building Blocks; Isotopic Labeled Analogues;
應(yīng)用:
Vernakalant-d6 Hydrochloride is the labeled analog of Vernakalant Hydrochloride(V128620), a novel, relatively atrial-selective antiarrhythmic drug that effectively and rapidly terminates atrial fibrillation (AF).
參考文獻(xiàn)
Mao, Z.L., et. al.: J. Clin. Pharmacol., 52, 1042 (2012); Mao, Z., et. al.: J. Pharmacokinet. Pharmacodynam., 38, 541 (2011)