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    歡迎光臨:萊耀標(biāo)準(zhǔn)品網(wǎng)!
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    LP-211
    產(chǎn)品基本信息
    產(chǎn)品編號(hào):L473405
    產(chǎn)品名稱:LP-211
    產(chǎn)品CAS:1052147-86-0
    規(guī)格含量:50mg
    產(chǎn)品價(jià)格:面議
    聯(lián)系我們:
    產(chǎn)品詳細(xì)介紹
    標(biāo)準(zhǔn)品編號(hào): L473405
    名稱: LP-211
    別名: 6-(4-([1,1'-Biphenyl]-2-yl)piperazin-1-yl)-N-(4-cyanobenzyl)hexanamide; 4-[1,1'-Biphenyl]-2-yl-N-[(4-cyanophenyl)methyl]-1-piperazinehexanamide
    CAS號(hào): 1052147-86-0
    分子式: C??H??N?O
    分子量: 466.62
    種類(lèi): Standards; Pharmaceutical/API Drug Impurities/Metabolites;
    應(yīng)用: LP-211 is a brain penetrant selective agonist for the serotonin 5-HT7 receptor used in pharmacological studies which showed that it underwent metabolic breakdown to RVIP(LA)7 and showed pharmacological activities such as induced hypothermia in mice and showed optimal pharmacokinetics in rats. LP-211 is also a drug analogue of piperazinehexanamide exhibiting 5-HT7 receptor affinity.
    參考文獻(xiàn)


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