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產(chǎn)品基本信息
產(chǎn)品編號(hào):S142903
產(chǎn)品名稱(chēng):Savolitinib
產(chǎn)品CAS:1313725-88-0
規(guī)格含量:5mg
產(chǎn)品價(jià)格:面議
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產(chǎn)品詳細(xì)介紹
標(biāo)準(zhǔn)品編號(hào):
S142903
名稱(chēng):
Savolitinib
別名:
Volitinib; 1-[(1S)-1-Imidazo[1,2-a]pyridin-6-ylethyl]-6-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,3-triazolo[4,5-b]pyrazine; AZD 6094; HM 5016504; HMPL 504
CAS號(hào):
1313725-88-0
分子式:
C??H??N?
外觀:
Pale Beige Solid
熔點(diǎn):
205-207°C
分子量:
345.36
儲(chǔ)存:
-20°C Freezer
溶解度:
DMSO (Slightly), Methanol (Slightly)
類(lèi)別:
Standards; Enzyme Activators and Inhibitors;
應(yīng)用:
Savolitinib is a potent and highly selective c-Met inhibitor. Savoltinib demonstrated anti-tumor efficacy in a panel of cMet-dysregulated gastric cancer PDX models. Savolitinib also demonstrated good antitmuor activities.
參考文獻(xiàn)
Gavine, P., et al.: Mol. Oncol., 9, 323 (2015); Jia, H., et al.: J. Med. Chem., 57, 7577 (2014);
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