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    歡迎光臨:萊耀標(biāo)準(zhǔn)品網(wǎng)!
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    Pracinostat
    產(chǎn)品基本信息
    產(chǎn)品編號(hào):P699100
    產(chǎn)品名稱:Pracinostat
    產(chǎn)品CAS:929016-96-6
    規(guī)格含量:100mg
    產(chǎn)品價(jià)格:面議
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    產(chǎn)品詳細(xì)介紹
    標(biāo)準(zhǔn)品編號(hào): P699100
    名稱: Pracinostat
    別名: (2E)-3-[2-Butyl-1-[2-(diethylamino)ethyl]-1H-benzimidazol-5-yl]-N-hydroxyacrylamide; (E)-3-[2-Butyl-1-(2-diethylaminoethyl)-1H-benzimidazol-5-yl]-N-hydroxy-2-propenamide; Kaempferol 3-O-β-D-(6-E-p-Coumaroylglucoside); SB 939; SB939; (2E)-3-[2-Butyl-1-[2-(diethylamino)ethyl]-1H-benzimidazol-5-yl]-N-hydroxy-2-propenamide;
    CAS號(hào): 929016-96-6
    分子式: C??H??N?O?
    分子量: 358.48
    類別: Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
    應(yīng)用: Pracinostat is a potent and orally active histone deacetylase (HDAC) inhibitor with high tumor exposure and efficacy in mouse models of colorectal cancer. The selectivity of Pracinostat for tumor tissues makes it a promising therapeutic candidate for use in patients with advanced solid malignancies. Potent Histone deacetylase inhibitor.
    參考文獻(xiàn)


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