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    Cariprazine-d8
    產(chǎn)品基本信息
    產(chǎn)品編號:C183492
    產(chǎn)品名稱:Cariprazine-d8
    產(chǎn)品CAS:1308278-69-4
    規(guī)格含量:10mg
    產(chǎn)品價格:面議
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    產(chǎn)品詳細(xì)介紹
    標(biāo)準(zhǔn)品編號: C183492
    名稱: Cariprazine-d8
    別名: N'-[trans-4-[2-[4-(2,3-Dichlorophenyl)-1-piperazinyl]ethyl-2,2-d2]cyclohexyl]-N,N-di(methyl-d3)-urea;
    CAS號: 1308278-69-4
    參考CAS: 未標(biāo)記:839712-12-8
    分子式: C??H??D?Cl?N?O
    分子量: 435.46
    類別: Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;
    應(yīng)用: Cariprazine-d8 is a deuterated cyclohexyl urea modulators of D2 receptors and/or modulators of D3 receptors for disease treatment in relation to increased enzymic metabolic stability. Also, it is derived from N-(2,3-Dichlorophenyl)piperazine-d8 (D435752), which is a compound useful in organic synthesis. A deuterated form of Cariprazine (C183490), which is an orally active D2/D3 dopamine receptor antagonist (1,2,3). Cariprazine is an antipsychotic drug candidate for the potential treatment of schizophrenia, bipolar mania and depression.
    參考文獻(xiàn)


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